
%0 Journal Article
%A Millan, David S. 
%A Prager, Rolf H. 
%T Potential GABA<emph type="8">B</emph> Receptor Antagonists. XI. Synthesis of a Small Library of Sulfonamide Analogues
%J Australian Journal of Chemistry
%D 2000/10/27
%V 53
%N 7
%P 615-618
%K Combinatorial synthesis; GABAB antagonists; heteroarylaminopropanesulfonamides; Rink resin.
%R https://doi.org/10.1071/CH00067
%U https://www.publish.csiro.au/paper/CH00067 
%X The synthesis of a small library of 3-heteroarylaminopropane-1-sulfonamide analogues of 4-aminobutanoic acid (GABA) by solid-phase chemistry is reported. None showed any significant activity as agonists or antagonists of GABAA or GABAB receptors in the guinea pig ileum. 
