
TY  - JOUR
A1  - Millan, David S. 
A1  - Prager, Rolf H. 
T1  - Potential GABA<emph type="8">B</emph> Receptor Antagonists. XI. Synthesis of a Small Library of Sulfonamide Analogues
JF  - Australian Journal of Chemistry
JO  - Aust. J. Chem.
Y1  - 2000
VL  - 53
IS  - 7
SP  - 615
EP  - 618
KW  - Combinatorial synthesis; GABAB antagonists; heteroarylaminopropanesulfonamides; Rink resin.
UR  - https://doi.org/10.1071/CH00067 
N2  - The synthesis of a small library of 3-heteroarylaminopropane-1-sulfonamide analogues of 4-aminobutanoic acid (GABA) by solid-phase chemistry is reported. None showed any significant activity as agonists or antagonists of GABAA or GABAB receptors in the guinea pig ileum. 
ER  -

